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- Antipsychotic Powder Trifluoperazine Dihydrochloride For Antiadrenergic Effects CAS:440-17-5
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- Product Name: Trifluoperazine Dihydrochloride
- Synonyms:10-[3-(4-Methyl-1-Piperazinyl)Propyl]-2-Trifluoromethyl-Phenothiazine Dihydrochloride;10-[3-(4-Methylpiperazin-1-Yl)Propyl]-2-(Trifluoromethyl)-10h-Phenothiazine Dihydrochloride;Stelazine;Stelazine Dihydrochloride;Trifluoperazine 2hcl;Trifluoperazine HCL
- CAS:440-17-5
- MF:C21H26Cl2F3N3S
- MW:480.42
- EINECS:207-123-0
- Melting point:243 °C (dec.)(lit.)
- Chemical Properties:Cream Fine Powder
- Usage: Antipsychotic.
- Trifluoperazine dihydrochloride
- Trifluoperazine Dihydrochloride is a cell-permeable phenothiazine compound with antiadrenergic effects. Trifluoperazine is described as an antagonist of adrenergic receptors, demonstrating much higher activity at the α-1 over the α-2 adrenergic receptor. Trifluoperazine is also described to produce antidopaminergic effects. Trifluoperazine facilitates agonist induced elevation of cytosolic calcium at low concentrations (10μM), and antagonizes CaM (calmodulin) at higher concentrations. Potent and irreversible inhibitor of cAMP-gated cationic channels. Inhibits DNA repair. Potent neurotoxin. Trifluoperazine is an inhibitor of D2DR.
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